Search Result "Radiolabeled P-gp substrates"


Substrates, Inhibitors and Activators of P-glycoprotein: Candidates for Radiolabeling and Imaging Perspectives

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1703-1714
Author(s): Nicola A. Colabufo, Francesco Berardi, Maria Grazia Perrone, Elena Capparelli, Mariangela Cantore, Carmela Inglese, Roberto Perrone

Review Article

Design and Synthesis of New Selective P-gp Substrates and Inhibitors

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5774-5778
Author(s): Mariangela Cantore,Marcello Leopoldo,Francesco Berardi,Roberto Perrone,Nicola Antonio Colabufo

Study of Oxidized Lipids as Endogenous Substrates of P-gp (ABCB1)

Journal: Drug Metabolism Letters
Volume: 2 Issue: 4 Year: 2008 Page: 238-244
Author(s): Masatoshi Masuda, Emi Nakai, Takaharu Mizutani

A New Method to Measure P-gp (ABCB1) Activity

Journal: Drug Metabolism Letters
Volume: 1 Issue: 4 Year: 2007 Page: 306-310
Author(s): Masatoshi Masuda, Takaharu Mizutani

11C-verapamil to Assess P-gp Function in Human Brain During Aging,Depression and Neurodegenerative Disease

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1775-1784
Author(s): A. L. Bartels, O. L. de Klerk, R. Kortekaas, J. J. de Vries, K. L. Leenders

Modulation and Absorption of Xenobiotics: The Synergistic Role of CYP450 and P-gp Activities in Cancer and Neurodegenerative Disorders

Journal: Current Drug Metabolism
Volume: 12 Issue: 8 Year: 2011 Page: 702-712
Author(s): Carmela Inglese, Maria Grazia Perrone, Francesco Berardi, Roberto Perrone, Nicola Antonio Colabufo

Using PET Studies of P-gp Function to Elucidate Mechanisms Underlying the Disposition of Drugs

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1799-1809
Author(s): Stina Syvanen, Margareta Hammarlund-Udenaes

Imaging Drug Resistance with Radiolabeled Molecules

Journal: Current Pharmaceutical Design
Volume: 10 Issue: 2 Year: 2004 Page: 2965-2979
Author(s): G. Vaidyanathan, M. R. Zalutsky

Loxapine P-glycoprotein Interactions In Vitro

Journal: Drug Metabolism Letters
Volume: 6 Issue: 1 Year: 2012 Page: 26-32
Author(s): Andrea Reed, Keith Huie, Elke S. Perloff, James V. Cassella, Lori H. Takahashi

Pharmacodynamics of Radiolabelled Anticancer Drugs for Positron Emission Tomography

Journal: Current Pharmaceutical Design
Volume: 9 Issue: 1 Year: 2003 Page: 931-944
Author(s): O. Clyde Hutchinson, David R. Collingridge, Henryk Barthel, Pat. M. Price, Eric O. Aboagye

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